Ac-DEVD-CHO
Lieferant: ENZO LIFE SCIENCES
ALX260030M001
ALX260030M005
ENZOALX260030M001EA
96.8
EUR
ENZOALX260030M001
ENZOALX260030M005
Ac-DEVD-CHO
Proteine und Peptide
Caspase-3 inhibitor
Highly specific, potent and reversible inhibitor of caspase-3. Ki<1 nM for purified caspase-3. IC50=0,2 nM for PARP cleavage in cultured human osteosarcoma cell extracts. In contrast, the caspase-1 (ICE) specific inhibitor YVAD-CHO has a Ki=12 µM for caspase-3 and IC50>10 µM for PARP cleavage in osteosarcoma cell extracts. The DEVD sequence is based on PARP cleavage site Asp-216 for caspase-3.
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